SCHEMBL8637899

SCHEMBL8637899

COc1cccc(Cc2nc(Cl)c(Oc3ccccc3OC)c(OS(=O)(=O)c3ccc(C(C)C)cn3)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHPS P49366 2/20 0.43
EDNRA P25101 18/20 0.43
EDNRB P24530 17/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635722 0.93 DHPS (0.35) DHPSEDNRAEDNRB
SCHEMBL8635760 0.89 DHPS (0.50) DHPSEDNRAEDNRB
SCHEMBL8631708 0.81 DHPS (0.42) DHPSEDNRAEDNRB
SCHEMBL7850977 0.77 DHPS (0.65) DHPS
SCHEMBL8638012 0.73 DHPS (0.39) DHPSEDNRAEDNRB
SCHEMBL8395334 0.73 LMNA (0.37) DHPSEDNRAEDNRB
SCHEMBL7852059 0.72 EDNRA (0.65) DHPSEDNRAEDNRB
SCHEMBL31037804 0.68 DHPS (0.66) DHPS
SCHEMBL7851037 0.68 DHPS (0.52) DHPS
SCHEMBL6785297 0.68 EDNRA (0.66) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5837708-A CARDIOVASCULAR DISORDERS OF HYPERTENSION, ISCHEMIA, ANGINA PECTORIS AND VASOSPASMS HOFFMANN-LA ROCHE INC. (US) 1998-11-17 US disclosed