SCHEMBL8635781

SCHEMBL8635781

COC(=O)Cc1cccc2c1Sc1c(C=O)cccc1N2C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 1/20 0.35
ERN1 O75460 1/20 0.35
TLR1 Q15399 1/20 0.35
TLR6 Q9Y2C9 1/20 0.35
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 5/20 0.33
POLB P06746 2/20 0.33
NFE2L2 Q16236 1/20 0.33
KDM1A O60341 1/20 0.33
RAB9A P51151 1/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 4/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32
PABPC1 P11940 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630372 0.87 USP2 (0.34) KDM4EALDH1A1POLBKDM1AMEN1
SCHEMBL8630374 0.87 USP2 (0.34) KDM4EALDH1A1POLBKDM1AMEN1
Hydrochloric Acid SCHEMBL8629084 0.82 CFD (0.38) KDM4EALDH1A1POLBKDM1AMEN1
SCHEMBL8632827 0.78 RIPK1 (0.36) KDM4EALDH1A1KDM1AKMT2AMAPT
SCHEMBL4893812 0.74 ALDH1A1 (0.44) TLR2ERN1TLR1TLR6KDM4E
SCHEMBL8633026 0.73 BACE1 (0.40)
SCHEMBL9011882 0.72 ALDH1A1 (0.43) TLR2ERN1TLR1TLR6KDM4E
SCHEMBL7392294 0.70 MAOA (0.56) KDM4EALDH1A1POLBRAB9AMEN1
SCHEMBL7429083 0.70 SMYD2 (0.30)
SCHEMBL7394096 0.69 ALDH1A1 (0.33) TLR2ERN1TLR1TLR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811548-A USEFUL AS RESEARCH TOOLS IN THE DETERMINATION OF BIOLOGICALLY ACTIVE PEPTIDE SEQUENCES HOFFMANN-LA ROCHE INC. (US) 1998-09-22 US disclosed
US-5811389-A INHIBITING PLATELET AGGREGATION; BLOOD DISORDERS HOFFMANN-LA ROCHE INC. (US) 1998-09-22 US disclosed