SCHEMBL8638848

SCHEMBL8638848

O=C1CC(=O)N(c2ccccc2)c2ccccc2N1CCC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 16/20 0.58
ALDH1A1 P00352 1/20 0.43
CASP7 P55210 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HPGD P15428 1/20 0.43
EPHX2 P34913 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619499 0.88 CCKBR (0.55) CCKBRHPGDEPHX2
SCHEMBL9436139 0.85 CCKBR (0.53) CCKBRHPGDEPHX2
SCHEMBL8638391 0.81 CCKBR (0.64) CCKBR
SCHEMBL8616285 0.80 CCKBR (0.46) CCKBRHPGDEPHX2
SCHEMBL7044712 0.76 HPGD (0.53) CCKBRALDH1A1HSD17B10HPGD
SCHEMBL8616731 0.76 CCKBR (0.51) CCKBRALDH1A1HSD17B10HPGD
SCHEMBL8639633 0.75 KMT2A (0.62) CCKBRALDH1A1CASP7HSD17B10HPGD
SCHEMBL8635136 0.74 NPC1 (0.52) CCKBRALDH1A1HSD17B10HPGD
SCHEMBL8635124 0.74 CCKBR (0.73) CCKBR
SCHEMBL4422153 0.73 HPGD (0.74) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558104-B1 1,5-Benzodiazepine derivatives and their use in medicine GLAXO WELLCOME SPA (IT) 1998-07-29 EP disclosed
US-5637697-A ANTAGONIST TO GASTRIN AND(OR) CHLOROCYSTOKININ GLAXO SPA (IT) 1997-06-10 US disclosed
US-5580895-A GASTROINTESTINAL OR CENTRAL NERVOUS SYSTEM DISORDERS GLAXO SPA (IT) 1996-12-03 US disclosed
EP-0558104-A1 1,5-Benzodiazepine derivatives and their use in medicine GLAXO S.p.A. (IT) 1993-09-01 EP disclosed