SCHEMBL8639006

SCHEMBL8639006

COc1ccc([C]=O)cc1C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.46
RARA P10276 2/20 0.43
RARB P10826 2/20 0.43
RARG P13631 2/20 0.43
CYP3A4 P08684 3/20 0.43
HPGD P15428 2/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
ALOX15 P16050 1/20 0.43
WDR5 P61964 1/20 0.39
ERBB2 P04626 2/20 0.38
HTR2A P28223 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
EGFR P00533 1/20 0.36
LPAR1 Q92633 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
CYP19A1 P11511 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3130927 0.85 CYP3A4 (0.43) ALDH1A1GAARARARARBRARG
SCHEMBL512996 0.84 ESRRB (0.40) ALDH1A1GAAHPGDHTR2APGR
SCHEMBL10211666 0.81 AR (0.49) ALDH1A1GAARARARARBRARG
SCHEMBL9350206 0.81 RXRA (0.35) ALDH1A1GAATDP1PTGDR2KMT2A
SCHEMBL18913771 0.78 RARA (0.48) ALDH1A1GAARARARARBRARG
SCHEMBL56335 0.78 CA2 (0.48) ALDH1A1GAACYP3A4HPGDTDP1
SCHEMBL9491535 0.76 CNR2 (0.44) CYP3A4LMNATP53ALOX15NR3C1
SCHEMBL6210745 0.75 AR (0.40) ALDH1A1CYP3A4HPGDLMNAALOX15
SCHEMBL11673151 0.75 ALDH1A1 (0.40) ALDH1A1CYP3A4HPGDTDP1CA1
SCHEMBL5680098 0.75 PTGS2 (0.42) ALDH1A1RARGCYP3A4HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661258-B1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CIRD GALDERMA (FR) 1998-04-08 EP disclosed
EP-0514264-B1 Biaromatic compounds derived from compounds having a salicylic configuration, their preparation process and their use in human and veterinary medicine and in cosmetics CIRD GALDERMA (FR) 1995-11-15 EP disclosed
EP-0514269-B1 Imino-derivatives, process for their preparation and their use in human and veterinary medicine and in cosmetics CIRD GALDERMA (FR) 1995-11-02 EP disclosed
EP-0661258-A1 Biaromatic propynyl compounds, pharmaceutical compositions and cosmetics containing them and their uses CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA, ( CIRD GALDERMA) (FR) 1995-07-05 EP disclosed
EP-0552282-B1 BI-AROMATIC COMPOUNDS AND THEIR USE IN HUMAN AND VETERINARY MEDECINE AND IN COSMETIC PREPARATIONS CIRD GALDERMA (FR) 1994-08-24 EP disclosed
EP-0552282-A1 BI-AROMATIC COMPOUNDS AND THEIR USE IN HUMAN AND VETERINARY MEDECINE AND IN COSMETIC PREPARATIONS. CIRD GALDERMA (FR) 1993-07-28 EP disclosed
WO-1992020643-A1 NOVEL BI-AROMATIC COMPOUNDS DERIVED FROM A SALICILIC PATTERN, METHOD OF PREPARATION AND USE IN HUMAN AND VETERINARY MEDECINE AND IN COSMETICS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (CIRD GALDERMA) (FR) 1992-11-26 WO disclosed
EP-0514269-A1 Imino-derivatives, process for their preparation and their use in human and veterinary medicine and in cosmetics CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA, ( CIRD GALDERMA) (FR) 1992-11-19 EP disclosed
EP-0514264-A1 Biaromatic compounds derived from compounds having a salicylic configuration, their preparation process and their use in human and veterinary medicine and in cosmetics CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA, ( CIRD GALDERMA) (FR) 1992-11-19 EP disclosed
WO-1992006948-A1 BI-AROMATIC COMPOUNDS AND THEIR USE IN HUMAN AND VETERINARY MEDECINE AND IN COSMETIC PREPARATIONS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (CIRD GALDERMA) (FR) 1992-04-30 WO disclosed