SCHEMBL8648902

SCHEMBL8648902

O=C(c1ccc(Cl)cc1)C(Cl)(Cl)Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.56
CES1 P23141 3/20 0.56
TSHR P16473 2/20 0.54
ALOX15 P16050 1/20 0.54
ALDH1A1 P00352 2/20 0.53
HPGD P15428 1/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
GSK3B P49841 2/20 0.48
MAPK1 P28482 2/20 0.48
SRD5A2 P31213 1/20 0.48
L3MBTL1 Q9Y468 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.42
ATM Q13315 1/20 0.42
PTGS2 P35354 1/20 0.42
ERCC5 P28715 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10620118 0.89 ALDH1A1 (0.41) CES2CES1TSHRALOX15ALDH1A1
SCHEMBL10662968 0.88 MMP1 (0.53) CES2CES1TSHRALOX15ALDH1A1
SCHEMBL10348275 0.82 RXRA (0.40) CES1ALDH1A1HPGDGSK3BL3MBTL1
SCHEMBL10405986 0.82 CES2 (0.59) CES2CES1TSHRALOX15ALDH1A1
SCHEMBL10887646 0.81 CES2 (0.52) CES2CES1TSHRALOX15ALDH1A1
SCHEMBL7532519 0.80 MAPT (0.52) CES2ALDH1A1HPGDCA1CA2
SCHEMBL19303575 0.78 CES2 (0.54) CES2CES1TSHRALOX15ALDH1A1
SCHEMBL8167899 0.78 CA2 (0.55) CES2CES1ALDH1A1HPGDCA2
SCHEMBL978677 0.78 CES1 (0.60) CES2CES1TSHRALOX15ALDH1A1
SCHEMBL17187854 0.78 CES2 (0.54) CES2CES1TSHRALOX15ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767314-A Selective acylation of monoalkylhydrazines ROHM AND HAAS COMPANY (US) 1998-06-16 US disclosed
US-5675037-A REACTING UNSUBSTITUTED OR MONOALKYL-HYDRAZINES WITH TRICHLOROMETHYL ARYL KETONES ROHM AND HAAS COMPANY (US) 1997-10-07 US disclosed
CN-1032254-C Selective acylation of hydrazines ROHM & HAAS (US) 1996-07-10 CN disclosed
EP-0492839-B1 Selective acylation of hydrazines ROHM & HAAS (US) 1995-04-12 EP disclosed