SCHEMBL8650329

SCHEMBL8650329

Cc1ccc(S(=O)(=O)OCCCc2csc3ccc(F)cc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.46
MTNR1B P49286 2/20 0.46
CA2 P00918 2/20 0.46
PSMD10 O75832 1/20 0.36
MAPT P10636 5/20 0.35
TP53 P04637 3/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
CYP24A1 Q07973 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
THRB P10828 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8646966 0.87 CA2 (0.46) MTNR1AMTNR1BCA2PSMD10MAPT
SCHEMBL8645804 0.84 SMN1; SMN2 (0.44) MTNR1ACA2PSMD10TP53CA12
SCHEMBL8788554 0.83 PSMD10 (0.41) MTNR1AMTNR1BCA2PSMD10
SCHEMBL4351623 0.78 MPO (0.54)
SCHEMBL8650318 0.78 THRB (0.39) MTNR1ACA2PSMD10MAPTCA12
SCHEMBL8649697 0.76 SMN1; SMN2 (0.46) MTNR1ACA2TP53CA12CA1
SCHEMBL9213281 0.76 HTR2A (0.48)
SCHEMBL16433177 0.75 MPO (0.55)
SCHEMBL4793354 0.74 FKBP1A (0.52) CA2PSMD10MAPTCA1
SCHEMBL8780822 0.72 ALDH1A1 (0.44) PSMD10CYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763444-A CENTRAL NERVOUS SYSTEM AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-06-09 US disclosed
EP-0761666-A2 Antidepressant 1-arylalkyl-4-(alkoxypyridinyl)- or 4-(alkoxypyrimidinyl)piperazine derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-12 EP disclosed