SCHEMBL8650343

SCHEMBL8650343

NC(=O)c1ccc2scc(CCCO)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 0.41
MTNR1B P49286 4/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
HTR1A P08908 2/20 0.39
HTR1D P28221 2/20 0.39
HTR2C P28335 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
TSHR P16473 1/20 0.39
HTR1B P28222 1/20 0.39
HTR7 P34969 1/20 0.39
HTR5A P47898 1/20 0.39
HTR6 P50406 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650374 0.85 CA2 (0.41) MTNR1AMTNR1B
SCHEMBL23612316 0.79 CYP2A6 (0.41) MTNR1AMTNR1BKEAP1NFE2L2HTR5A
SCHEMBL8788477 0.77 MTNR1A (0.38) MTNR1AMTNR1BKEAP1NFE2L2HTR1A
SCHEMBL8653030 0.76 CYP2A6 (0.61) MTNR1AMTNR1BKEAP1NFE2L2HDAC10
SCHEMBL8648779 0.76 MTNR1A (0.58) MTNR1AMTNR1BKEAP1NFE2L2CYP2A6
SCHEMBL8788554 0.75 PSMD10 (0.41) MTNR1AMTNR1B
SCHEMBL8255715 0.72 CYP2A6 (0.42) MTNR1AMTNR1BKEAP1NFE2L2HTR1A
SCHEMBL14155053 0.72 CA2 (0.49) MTNR1AMTNR1BKEAP1NFE2L2CYP2A6
SCHEMBL79170 0.72 CYP2A6 (0.69) MTNR1AHDAC6CYP2A6
SCHEMBL27989610 0.71 HTR7 (0.74) HTR1AHTR1DHTR2CMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763444-A CENTRAL NERVOUS SYSTEM AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-06-09 US disclosed
EP-0761666-A2 Antidepressant 1-arylalkyl-4-(alkoxypyridinyl)- or 4-(alkoxypyrimidinyl)piperazine derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-12 EP disclosed