SCHEMBL8788477

SCHEMBL8788477

CC(C)(C)[Si](C)(C)OCCCc1csc2ccc(C(N)=O)cc12

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 12/20 0.38
MTNR1B P49286 7/20 0.38
HTR1A P08908 2/20 0.36
HTR1D P28221 2/20 0.36
HTR2C P28335 2/20 0.36
KIF11 P52732 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8789180 0.81 CYP2A6 (0.48) MTNR1AMTNR1B
SCHEMBL8650343 0.77 MTNR1A (0.41) MTNR1AMTNR1BHTR1AHTR1DHTR2C
SCHEMBL8788554 0.74 PSMD10 (0.41) MTNR1AMTNR1BKIF11HRH3
SCHEMBL22937053 0.70 TSHR (0.42) HRH3
SCHEMBL29686890 0.69 PRSS1 (0.50) HTR1A
SCHEMBL8650374 0.68 CA2 (0.41) MTNR1AMTNR1BKIF11HRH3
SCHEMBL22937051 0.66 RARG (0.39)
SCHEMBL28752006 0.66 PRSS1 (0.46)
SCHEMBL29686658 0.66 PRSS1 (0.46)
SCHEMBL29170120 0.65 ALDH1A1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0761666-A2 Antidepressant 1-arylalkyl-4-(alkoxypyridinyl)- or 4-(alkoxypyrimidinyl)piperazine derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-12 EP disclosed