SCHEMBL8658246

SCHEMBL8658246

O=c1[nH]c(-c2ccccc2)cn1-n1cc(-c2ccsc2)[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.47
CYP2A6 P11509 1/20 0.47
CYP2B6 P20813 1/20 0.47
GLO1 Q04760 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ERCC1 P07992 1/20 0.41
FEN1 P39748 1/20 0.41
ERCC4 Q92889 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
NPY5R Q15761 1/20 0.39
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 2/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8406497 0.85 ERCC1 (0.52) SMN1; SMN2ERCC1FEN1ERCC4CA12
SCHEMBL8518603 0.83 GLO1 (0.40) CYP2E1CYP2A6CYP2B6GLO1SMN1; SMN2
SCHEMBL8660223 0.81 CYP2E1 (0.36) CYP2E1CYP2A6CYP2B6GLO1SMN1; SMN2
SCHEMBL8987160 0.70 CYP2E1 (0.53) CYP2E1CYP2A6CYP2B6GLO1SMN1; SMN2
SCHEMBL5935431 0.70 KMT2A (0.48) SMN1; SMN2ERCC1FEN1ERCC4CA12
SCHEMBL4736133 0.68 RAB9A (0.69) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL9880650 0.67 ERCC1 (0.49) SMN1; SMN2ERCC1FEN1ERCC4CA12
SCHEMBL13806371 0.67 CA12 (0.50) SMN1; SMN2ERCC1FEN1ERCC4CA12
SCHEMBL14417266 0.67 DRD2 (0.43) DRD2DRD4DRD3CCNB2CDK1
SCHEMBL149952 0.67 CYP2A6 (1.00) CYP2E1CYP2A6CYP2B6GLO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927192-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1999-07-07 EP claimed
WO-1998011128-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1998-03-19 WO claimed