SCHEMBL8660223

SCHEMBL8660223

O=C1[N]C(c2ccccc2)=CN1n1cc(-c2ccsc2)[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2B6 P20813 1/20 0.36
GLO1 Q04760 1/20 0.33
KDM4E B2RXH2 2/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPY5R Q15761 1/20 0.32
FYN P06241 1/20 0.32
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CCNB2 O95067 1/20 0.30
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
GSK3B P49841 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560492 0.88 ERCC1 (0.38) KDM4EHSD17B10NPY5RALDH1A1HPGD
SCHEMBL8658246 0.81 CYP2E1 (0.47) CYP2E1CYP2A6CYP2B6GLO1KDM4E
SCHEMBL8518603 0.71 GLO1 (0.40) CYP2E1CYP2A6CYP2B6GLO1KDM4E
SCHEMBL8406497 0.67 ERCC1 (0.52) KDM4ENPSR1HSD17B10ALDH1A1HPGD
SCHEMBL8987160 0.60 CYP2E1 (0.53) CYP2E1CYP2A6CYP2B6GLO1KDM4E
SCHEMBL4736133 0.58 RAB9A (0.69) KDM4EALDH1A1POLBHPGDSMN1; SMN2
SCHEMBL14417266 0.58 DRD2 (0.43) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL5935431 0.57 KMT2A (0.48) KDM4EHSD17B10NPY5RALDH1A1HPGD
SCHEMBL149952 0.57 CYP2A6 (1.00) CYP2E1CYP2A6CYP2B6GLO1FYN
SCHEMBL13801337 0.57 DRD2 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927192-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1999-07-07 EP disclosed
WO-1998011128-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1998-03-19 WO disclosed