SCHEMBL8664832

SCHEMBL8664832

[c]1scc(-c2ccccc2)c1-c1ccccc1N1CCOCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.43
HTR1A P08908 1/20 0.43
HTR7 P34969 1/20 0.43
HTR5A P47898 1/20 0.43
HTR6 P50406 1/20 0.43
AR P10275 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
PDE4A P27815 1/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 2/20 0.41
HSD17B10 Q99714 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
PIK3CD O00329 4/20 0.39
PIK3CA P42336 4/20 0.39
PIK3CB P42338 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664016 0.82 KMT2A (0.43) ARNPC1RAB9AMEN1MAPT
SCHEMBL8997930 0.82 MAPT (0.43) NPC1RAB9AMEN1MAPTKMT2A
SCHEMBL8665476 0.82 ALDH1A1 (0.43) ARNPC1RAB9AMEN1MAPT
SCHEMBL15362290 0.81 HTR7 (0.62) HTR2AHTR1AHTR7HTR5AHTR6
SCHEMBL8664502 0.79 AR (0.47) ARNPC1RAB9APDE4AMAPT
SCHEMBL8997879 0.78 MAPT (0.43) ARNPC1RAB9AMEN1MAPT
SCHEMBL8663981 0.73 PDE4A (0.42) HTR2AHTR1AHTR7HTR5AHTR6
SCHEMBL17628666 0.70 NPC1 (0.44) HTR7ARNPC1RAB9AMEN1
SCHEMBL9424119 0.68 LMNA (0.62) NPC1RAB9APDE4AMEN1MAPT
SCHEMBL21788597 0.67 SMN1; SMN2 (0.59) ARNPC1PDE4AMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852006-A N-aminoalkyl-substituted nitrogen-containing six membered heterocyclic compounds NIPPON CHEMIPHAR CO., LTD. (JP) 1998-12-22 US disclosed
US-5574030-A INHIBITING URINARY CONTRACTION, HETEROCYCLIC DIAMINES NIPPON CHEMIPHAR CO., LTD. (JP) 1996-11-12 US disclosed