SCHEMBL8666520

SCHEMBL8666520

CC(C)OC1=Nc2ccc(C#Cc3ccccc3C(=O)O)cc2C(C)(C)C1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RARB P10826 11/20 0.38
RARG P13631 11/20 0.38
RARA P10276 9/20 0.38
CYP26A1 O43174 2/20 0.35
CYP3A4 P08684 2/20 0.35
CRABP2 P29373 1/20 0.35
FFAR1 O14842 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HNF4A P41235 1/20 0.32
CXCR5 P32302 1/20 0.32
ALDH1A1 P00352 2/20 0.31
SLC6A9 P48067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633708 0.92 RARB (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8605739 0.85 RARB (0.53) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8605748 0.77 RARB (0.45) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8604136 0.76 RARB (0.53) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8580705 0.73 RARB (0.65) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8605671 0.69 RARB (0.43) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8633713 0.69 RARB (0.33) RARBRARGRARA
SCHEMBL27304274 0.68 RARB (0.62) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8772626 0.66 RARA (0.62) RARBRARGRARA
SCHEMBL8772741 0.66 RARA (0.53) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825986-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1998-03-04 EP disclosed
WO-1996036609-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-11-21 WO disclosed