SCHEMBL8670561

SCHEMBL8670561

Cn1nc(Cl)n(-c2ccc(Cl)cc2COS(C)(=O)=O)c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 2/20 0.35
SETDB1 Q15047 1/20 0.34
BRD9 Q9H8M2 1/20 0.33
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA1 P14867 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRA4 P48169 1/20 0.32
GABRA6 Q16445 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
BRD4 O60885 2/20 0.31
GALR3 O60755 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
ADORA2A P29274 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664376 0.89 SMN1; SMN2 (0.33) SETDB1BRD9SMN1; SMN2ALDH1A1LMNA
SCHEMBL8666669 0.85 SETDB1 (0.36) SETDB1SMN1; SMN2BRD4CYP1A2CYP3A4
SCHEMBL8664792 0.81 SETDB1 (0.42) SETDB1SMN1; SMN2GALR3CYP1A2CYP3A4
SCHEMBL8660658 0.80 SETDB1 (0.39) SETDB1BRD9GABRG2GABRB3GABRA5
SCHEMBL6487678 0.71 TRPV4 (0.39) DDR1ALDH1A1
SCHEMBL15413757 0.70 PSEN1 (0.41) DDR1SMN1; SMN2NPSR1LMNA
SCHEMBL2548023 0.68 NOS3 (0.38) DDR1HTTTSHRLMNA
SCHEMBL16550662 0.68 IDO1 (0.55) SMN1; SMN2CYP1A2CYP3A4CYP2C19HTT
SCHEMBL8675983 0.68 SETDB1 (0.38) SETDB1BRD9SMN1; SMN2HTTTSHR
SCHEMBL15415062 0.67 TRPV4 (0.50) SMN1; SMN2CYP1A2HTTTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874831-A1 PROCESSES AND COMPOUNDS FOR PREPARING CYCLIC UREA FUNGICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-11-04 EP disclosed
WO-1997019935-A1 PROCESSES AND COMPOUNDS FOR PREPARING CYCLIC UREA FUNGICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1997-06-05 WO disclosed