SCHEMBL8671302

SCHEMBL8671302

C#COC(=O)c1ccc(-c2ccc3c(c2)C(C)(C)CCC3=O)cc1CC

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PGR P06401 5/20 0.38
HSD17B1 P14061 3/20 0.37
RXRA P19793 4/20 0.34
RARG P13631 9/20 0.33
RARA P10276 7/20 0.33
RARB P10826 6/20 0.33
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9089192 0.84 PGR (0.32) PGRHSD17B1RXRARARGRARA
SCHEMBL8670891 0.84 PGR (0.44) PGRRXRARARGRARARARB
SCHEMBL8668855 0.79 RXRA (0.34) PGRHSD17B1RXRARARGRARA
SCHEMBL8671303 0.78 NPC1 (0.39) PGRRARGRARARARB
SCHEMBL8866201 0.77 HDAC3 (0.39) PGRHSD17B1RARGRARB
SCHEMBL9116437 0.76 HSD17B1 (0.35) PGRHSD17B1RARGRARARARB
SCHEMBL8670887 0.75 PGR (0.39) PGRRXRARARGRARARARB
SCHEMBL8772692 0.72 RARB (0.45) RXRARARGRARARARBRXRB
SCHEMBL9425658 0.70 HSD17B1 (0.43) HSD17B1RXRARXRBRXRG
SCHEMBL13613860 0.68 CYP26A1 (0.37) PGRHSD17B1RXRARARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723620-A Acetylenes disubstituted with a 5 substituted tetrahydronaphthyl group and with an aryl or heteroaryl groups having retinoid-like biological activity ALLERGAN (US) 1998-03-03 US disclosed