SCHEMBL9116437

SCHEMBL9116437

C#COC(=O)c1ccc(-c2ccc3c(c2)C(C)(C)CC(=O)O3)cc1CC

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.35
PGR P06401 4/20 0.32
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8866201 0.80 HDAC3 (0.39) HSD17B1PGRRARBRARG
SCHEMBL9023693 0.79 NPC1 (0.36) RARARARBRARGKDM4EALDH1A1
SCHEMBL8671302 0.76 PGR (0.38) HSD17B1PGRRARARARBRARG
SCHEMBL9024438 0.75 RARA (0.38) PGRRARARARBRARGKDM4E
SCHEMBL9024949 0.75 NPC1 (0.45) RARARARBRARGKDM4EALDH1A1
SCHEMBL8668855 0.74 RXRA (0.34) HSD17B1PGRRARARARBRARG
SCHEMBL9425658 0.72 HSD17B1 (0.43) HSD17B1
SCHEMBL9116297 0.71 JAK2 (0.36) KDM4EALDH1A1HPGD
SCHEMBL8564690 0.71 RARA (0.43) RARARARBRARGKDM4EALDH1A1
SCHEMBL9089192 0.70 PGR (0.32) HSD17B1PGRRARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995018803-A1 ACETYLENES DISUBSTITUTED WITH A PHENYL OR HETEROARYL GROUP AND A 2-OXOCHROMANYL, 2-OXOTHIOCHROMANYL OR 2-OXO-1,2,3,4-TETRAHYDROQUINOLINYL GROUP HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1995-07-13 WO disclosed