SCHEMBL8698491

SCHEMBL8698491

CCOC(=O)C(C)(c1cc(C)cc(C)c1)C(c1ccc2[nH]ccc2c1)C(C)(N)C(CCCCc1ccncc1)C(=O)OCc1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.33
NR3C1 P04150 1/20 0.32
GNRHR P30968 7/20 0.31
F2 P00734 1/20 0.31
F10 P00742 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8698458 0.79 ENPP2 (0.38) ENPP2NR3C1GNRHRSLC6A2SLC6A4
SCHEMBL8689640 0.69 MAOA (0.36) NR3C1SLC6A2SLC6A4SLC6A3CCNC
SCHEMBL8697815 0.67 PTGS2 (0.36) NR3C1SLC6A2SLC6A4SLC6A3CCNC
SCHEMBL8695280 0.64 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3
SCHEMBL2301833 0.59 SLC6A2 (0.54) ENPP2NR3C1SLC6A2SLC6A4SLC6A3
SCHEMBL27608010 0.58 ENPP2 (0.53) ENPP2SLC6A2SLC6A4SLC6A3HDAC1
SCHEMBL27742085 0.57 SLC6A2 (0.46) ENPP2F10SLC6A2SLC6A4SLC6A3
SCHEMBL10830196 0.56 ENPP2 (0.46) ENPP2F2HDAC1HDAC8
SCHEMBL28154516 0.56 MMP8 (0.52) SLC6A2SLC6A3
SCHEMBL188098 0.56 ENPP2 (0.60) ENPP2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780437-A ADMINISTERING TO TREAT SEX-HORMONE RELATED DISORDERS MERCK & CO., INC. (US) 1998-07-14 US disclosed