SCHEMBL8699461

SCHEMBL8699461

CCCCN(C(=C[N+](=O)[O-])NC)c1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.38
KCNN4 O15554 1/20 0.36
KCNA5 P22460 1/20 0.36
S1PR1 P21453 7/20 0.36
HTT P42858 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
VCP P55072 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP2C19 P33261 1/20 0.34
GPX4 P36969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7669449 0.81 MAPT (0.34) LMNAGPX4
SCHEMBL7668595 0.79 GAA (0.40) TRPV1KCNA5HTTGAAHPGD
SCHEMBL7670861 0.75 CHRNB2 (0.41) KCNA5HTTHPGDLMNA
SCHEMBL7666573 0.74 ALDH1A1 (0.36) LMNACYP3A4CYP2C9CYP2C19
SCHEMBL9800218 0.73 FAAH (0.47) TRPV1HTTLMNA
SCHEMBL9800223 0.73 FAAH (0.47) TRPV1HTTLMNA
SCHEMBL7669223 0.72 CHRNA7 (0.49) HTTGAALMNA
SCHEMBL7669029 0.72 CHRNB2 (0.46) KCNA5HTTHPGDLMNA
SCHEMBL7669230 0.72 CHRNA7 (0.49) HTTGAALMNA
SCHEMBL9718704 0.71 RIPK1 (0.47) HTTGAAHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849768-A α-unsaturated amines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-15 US disclosed