SCHEMBL8700474

SCHEMBL8700474

O=C1OC(=O)C(c2ccc3c(c2)OCO3)=C1c1ccc(Cl)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.77
EDNRA P25101 2/20 0.50
EDNRB P24530 1/20 0.50
CNR1 P21554 1/20 0.50
ALOX5 P09917 1/20 0.48
PTPRC P08575 1/20 0.47
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
MAP2K4 P45985 1/20 0.45
DYRK1A Q13627 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
MAOB P27338 1/20 0.44
MAPT P10636 5/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6316764 0.90 PTGS2 (0.87) PTGS2EDNRAEDNRBALOX5PTPRC
SCHEMBL4751583 0.87 PTGS2 (1.00) PTGS2EDNRAEDNRBALOX5PTPRC
SCHEMBL27765776 0.79 CNR1 (0.56) PTGS2CNR1ALOX5PTPRCNPC1
SCHEMBL8853342 0.77 EDNRA (0.58) PTGS2EDNRAEDNRB
SCHEMBL4789136 0.72 PTGS2 (0.72) PTGS2EDNRAEDNRBPTPRCNPC1
SCHEMBL29826933 0.71 MAOB (0.56) NPC1RAB9AMAP2K4MAOBMAPT
SCHEMBL409478 0.71 MAOB (0.56) NPC1RAB9AMAP2K4MAOBMAPT
SCHEMBL6675332 0.70 MEN1 (0.43) PTGS2KMT2AMEN1HPGDTNKS
SCHEMBL6429372 0.69 SMN1; SMN2 (0.57) MAPTKDM4EALDH1A1SMN1; SMN2TP53
SCHEMBL14882034 0.69 GAPDH (0.65) ALOX5NPC1RAB9AMAOBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998041521-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-09-24 WO disclosed