SCHEMBL8702736

SCHEMBL8702736

Cc1ccc(C(C)(C)C)c(SC2C(=O)OC(CCc3ccccc3)(c3ccccc3)CC2(O)OCCN2CCOCC2)c1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KIF11 P52732 1/20 0.33
KCNH2 Q12809 1/20 0.33
MEN1 O00255 5/20 0.32
KMT2A Q03164 5/20 0.32
TRPV4 Q9HBA0 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
ABCB1 P08183 1/20 0.32
SIGMAR1 Q99720 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
CYP2C19 P33261 1/20 0.31
PRCP P42785 1/20 0.31
TMEM97 Q5BJF2 1/20 0.31
F2R P25116 1/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696790 0.92 KDM4E (0.31) ALDH1A1MEN1KMT2A
SCHEMBL8697348 0.88
SCHEMBL8010688 0.73 LTA4H (0.39) ALDH1A1
SCHEMBL7999278 0.66 LTA4H (0.39) ALDH1A1MEN1KMT2A
SCHEMBL7758845 0.66 LDHA (0.48)
SCHEMBL8008735 0.64 KCNA5 (0.37) ALDH1A1SIGMAR1PKM
SCHEMBL8008687 0.61 LDHA (0.41)
SCHEMBL8010782 0.59 LDHA (0.38) L3MBTL1
SCHEMBL8341901 0.59 ALDH1A1 (0.38) ALDH1A1KCNH2MEN1KMT2ACYP3A4
SCHEMBL7074874 0.59 KDM4E (0.35) ALDH1A1MEN1KMT2AL3MBTL1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834506-A TREATMENT OF HIV, AIDS; ANTIVIRAL ACTIVITY IMPROVED BY JUDICIOUS PLACEMENT OF POLAR SUBSTITUENTS WARNER-LAMBERT COMPANY (US) 1998-11-10 US claimed
US-5834506-A TREATMENT OF HIV, AIDS; ANTIVIRAL ACTIVITY IMPROVED BY JUDICIOUS PLACEMENT OF POLAR SUBSTITUENTS WARNER-LAMBERT COMPANY (US) 1998-11-10 US disclosed