SCHEMBL8705691

SCHEMBL8705691

CC(C)(C)c1ccc(S(=O)(=O)NC(=O)C(Cc2ccccc2)c2ccc3nsnc3c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.50
ALDH1A1 P00352 1/20 0.50
ITGB3 P05106 1/20 0.45
ITGAV P06756 1/20 0.45
NLRP3 Q96P20 1/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
IKBKB O14920 1/20 0.39
EEF2K O00418 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 2/20 0.39
NR1I2 O75469 1/20 0.38
ADCY6 O43306 1/20 0.38
ADCY3 O60266 1/20 0.38
ADCY9 O60503 1/20 0.38
ADCY5 O95622 1/20 0.38
ADCY8 P40145 1/20 0.38
GCGR P47871 1/20 0.38
ADCY7 P51828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709132 0.92 EPHX2 (0.41) MAPTALDH1A1ITGB3ITGAVNLRP3
SCHEMBL8704794 0.92 ALDH1A1 (0.43) MAPTALDH1A1ITGB3ITGAVNLRP3
SCHEMBL8710102 0.92 EPHX2 (0.42) MAPTALDH1A1ITGB3ITGAVMEN1
SCHEMBL8705303 0.91 MAPT (0.40) MAPTALDH1A1ITGB3ITGAVMEN1
SCHEMBL8709538 0.91 NR1H4 (0.42) MAPTALDH1A1ITGB3ITGAVNLRP3
SCHEMBL8709447 0.91 ITGB3 (0.48) MAPTALDH1A1ITGB3ITGAVMEN1
SCHEMBL8709894 0.91 FLT1 (0.44) MAPTALDH1A1ITGB3ITGAVMEN1
SCHEMBL8706028 0.91 MAPT (0.41) MAPTALDH1A1ITGB3ITGAVNLRP3
SCHEMBL8709625 0.90 NLRP3 (0.43) MAPTALDH1A1ITGB3ITGAVNLRP3
SCHEMBL8709556 0.89 MEN1 (0.43) MAPTALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998041515-A1 ENDOTHOLIN RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-09-24 WO disclosed