SCHEMBL5598985

SCHEMBL5598985

CC(C)C(=O)[C@@H]1N(CCc2ccccc2)c2ccccc2C12CCNCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CACNA1G O43497 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
BCHE P06276 5/20 0.35
ACHE P22303 2/20 0.35
SIGMAR1 Q99720 3/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
OPRM1 P35372 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599554 0.82 MTNR1A (0.36) MTNR1AHDAC1HDAC6CACNA1GCACNA1H
SCHEMBL5599732 0.75 SMN1; SMN2 (0.38) HTR2AALDH1A1MAPTOPRM1
SCHEMBL5779471 0.71 POLB (0.37) MAPT
SCHEMBL5592351 0.68 HDAC1 (0.42) HDAC1HDAC6ALDH1A1OPRM1KCNH2
SCHEMBL8707482 0.67 HTR2C (0.38) HTR2CMAPK1
SCHEMBL1670310 0.65 HTR2C (0.49) CACNA1GCACNA1HCACNA1IHTR2CMAPK1
SCHEMBL6649033 0.64 HTR2C (0.40) HTR2CMAPK1
SCHEMBL5778898 0.63 FKBP1A (0.42) CACNA1GCACNA1HCACNA1IBCHEALDH1A1
SCHEMBL2801668 0.63 NOTUM (0.40) SIGMAR1MAPK1OPRM1
SCHEMBL14713128 0.63 SIGMAR1 (0.36) SIGMAR1HTR2AHTR2CUSP2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed