SCHEMBL8713586

SCHEMBL8713586

Cc1nc2cccc3n(CCCC4CCN(C(=O)C(F)(F)F)CC4)c(=O)c1n23

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.35
CNR2 P34972 1/20 0.34
NPY1R P25929 5/20 0.33
RIPK1 Q13546 1/20 0.33
HTR2C P28335 1/20 0.33
DRD2 P14416 2/20 0.33
HTR1A P08908 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
AKR1C3 P42330 1/20 0.32
RBP4 P02753 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717917 0.95 KDM1A (0.34) KDM1ACNR2RIPK1HTR2CDRD2
SCHEMBL8713342 0.93 DRD2 (0.34) NPY1RDRD2HTR1ADRD4DRD3
SCHEMBL8713886 0.88 HTR1A (0.34) HTR2CDRD2HTR1ADRD4DRD3
SCHEMBL8712463 0.86 GPR119 (0.43)
SCHEMBL7871606 0.81 GPR119 (0.45) ALDH1A1
Hydrochloric Acid SCHEMBL8716168 0.80 NPY1R (0.40) NPY1R
SCHEMBL8718329 0.78 ALDH1A1 (0.33) CNR2DRD2HTR1AALDH1A1TSHR
Hydrochloric Acid SCHEMBL7872294 0.77 ALDH1A1 (0.33) CNR2DRD2HTR1AALDH1A1TSHR
SCHEMBL7868688 0.77 ALDH1A1 (0.37) DRD2HTR1ADRD4ALDH1A1
SCHEMBL7868708 0.76 GPR119 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826686-A2 Tricyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-04 EP disclosed