SCHEMBL8713644

SCHEMBL8713644

N#Cc1cnn(-c2ccccc2)c1S(=O)(=O)c1cccc(C(=O)NC(N)=O)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 6/20 0.49
PTGS2 P35354 6/20 0.49
XDH P47989 2/20 0.39
EGFR P00533 2/20 0.39
FGFR1 P11362 2/20 0.39
KDR P35968 2/20 0.39
HSD17B10 Q99714 1/20 0.38
GRM5 P41594 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
GFER P55789 1/20 0.37
KAT6A Q92794 3/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7456055 0.67 MAOA (0.49) HSD17B10CA1CA2
SCHEMBL8551482 0.66 PTGS2 (0.46) PTGS1PTGS2XDHGFER
SCHEMBL4173369 0.65 PTGS1 (0.60) PTGS1PTGS2NPC1RAB9AGFER
SCHEMBL8551424 0.64 PTGS1 (0.65) PTGS1PTGS2XDHGFERCA12
SCHEMBL1613646 0.64 XDH (0.71) PTGS1PTGS2XDHNPC1RAB9A
SCHEMBL10773308 0.63 KMT2A (0.62) PTGS1PTGS2XDHHSD17B10NPC1
SCHEMBL13601056 0.61 KMT2A (0.69)
SCHEMBL40525 0.61 ALDH1A1 (0.69) HSD17B10NPC1RAB9ACA12CA1
Benzene SCHEMBL28074647 0.61 ALDH1A1 (0.69) HSD17B10NPC1RAB9ACA12CA1
SCHEMBL28166896 0.61 ALDH1A1 (0.69) HSD17B10NPC1RAB9ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-10007658-A None JP disclosed
JP-H107658-A DERIVATIVE OF SULFONYL UREIDOPYRAZOLE SUMITOMO PHARMACEUT CO LTD 1998-01-13 JP disclosed