SCHEMBL8713847

SCHEMBL8713847

O=C(O)c1cc2c3ccccc3n(Cc3ccccc3)c2nc1N1CCOCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.48
PKM P14618 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
POLB P06746 1/20 0.46
PIK3C2B O00750 3/20 0.44
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CA P42336 1/20 0.43
PIK3CB P42338 1/20 0.43
EGLN1 Q9GZT9 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
RAB9A P51151 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
DPP4 P27487 1/20 0.41
HPGD P15428 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712545 0.88 RXFP1 (0.54) PRKDCPKMNPSR1POLBALDH1A1
SCHEMBL8711984 0.77 ALDH1A1 (0.55) PKMNPSR1ALDH1A1KDM4ERXFP1
SCHEMBL8711799 0.77 CYP19A1 (0.48) PRKDCPKMNPSR1POLBALDH1A1
SCHEMBL400114 0.72 KDM4E (0.56) NPSR1ALDH1A1KDM4EHDAC1HDAC6
SCHEMBL13752240 0.70 PRKDC (0.57) PRKDCPOLBALDH1A1KDM4EPIK3CD
SCHEMBL4220258 0.70 PKM (0.60) PKMPOLBALDH1A1KDM4EPIK3CA
SCHEMBL9584516 0.69 POLB (0.51) PRKDCPOLBALDH1A1HDAC1HDAC11
SCHEMBL8387165 0.68 KMT2A (0.55) PRKDCPOLBALDH1A1KDM4EHDAC1
SCHEMBL6902224 0.67 CCR2 (0.67) PRKDCPOLBPIK3C2BALDH1A1KDM4E
SCHEMBL398278 0.67 TSHR (0.53) POLBALDH1A1KDM4EHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842176-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1998-05-20 EP claimed
WO-1997005137-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1997-02-13 WO claimed
EP-0842176-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1998-05-20 EP disclosed
WO-1997005137-A1 HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1997-02-13 WO disclosed