SCHEMBL8716367

SCHEMBL8716367

CCC(C)NC1=Nc2sccc2SN1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
HSP90AA1 P07900 1/20 0.36
CYP3A4 P08684 1/20 0.36
THRB P10828 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
CASP1 P29466 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
ELANE P08246 2/20 0.32
HCAR3 P49019 1/20 0.32
GAA P10253 1/20 0.30
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8478113 0.71 ALDH1A1 (0.33) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL8715972 0.69 ALDH1A1 (0.31) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL8721026 0.67 ALDH1A1 (0.33) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL8715780 0.64 HCAR3 (0.33) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL4695990 0.60 FDPS (0.47) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL13574526 0.60 FDPS (0.47) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL3028445 0.59 ALDH1A1 (0.45) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL49805 0.56 ALDH1A1 (1.00) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL7999039 0.54 ALDH1A1 (0.35) ALDH1A1TP53HSP90AA1CYP3A4THRB
SCHEMBL18647882 0.53 L3MBTL1 (0.47) ALDH1A1TP53HSP90AA1CYP3A4THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876379-A1 FUSED 1,2,4-THIADIAZINE AND FUSED 1,4-THIAZINE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1998-11-11 EP disclosed
WO-1997026265-A1 FUSED 1,2,4-THIADIAZINE AND FUSED 1,4-THIAZINE DERIVATIVES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1997-07-24 WO disclosed