SCHEMBL8716900

SCHEMBL8716900

COc1ccc2c[c]ccc2c1C(C)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 4/20 0.48
NCEH1 Q6PIU2 1/20 0.41
MAPK1 P28482 2/20 0.37
GAA P10253 2/20 0.37
LMNA P02545 3/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CYP3A4 P08684 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
USP2 O75604 1/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 2/20 0.34
MEN1 O00255 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717429 0.84 CA9 (0.35) CA9LMNACA12CA1CA7
SCHEMBL30676839 0.77 NCEH1 (0.65) CA9NCEH1LMNACYP3A4SMN1; SMN2
SCHEMBL3357585 0.77 NCEH1 (0.65) CA9NCEH1LMNACYP3A4SMN1; SMN2
SCHEMBL9739745 0.75 MAPT (0.40) MAPK1LMNACYP3A4MAPTKDM4E
SCHEMBL9164412 0.75 MAPT (0.36) NCEH1GAAMAPTKDM4EALDH1A1
SCHEMBL15410676 0.74 ALDH1A1 (0.36) MAPK1LMNACYP3A4SMN1; SMN2MAPT
SCHEMBL4326638 0.73 CYP19A1 (0.41) NCEH1CYP3A4SMN1; SMN2MAPTMEN1
SCHEMBL8722679 0.73 MAPT (0.35) NCEH1MAPTHPGD
SCHEMBL8556354 0.73 MAPT (0.35) CYP3A4MAPT
SCHEMBL4465114 0.73 CYP19A1 (0.41) NCEH1MAPK1LMNASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763455-A SEROTONIN RECEPTOR ANTAGONISTS WAKE FOREST UNIVERSITY (US) 1998-06-09 US disclosed
US-5760055-A PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS WAKE FOREST UNIVERSITY (US) 1998-06-02 US disclosed