SCHEMBL8717153

SCHEMBL8717153

O=[C]N(C(=O)CCc1ccccc1)N1CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.42
SIGMAR1 Q99720 3/20 0.42
NPC1 O15118 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
SLC6A4 P31645 1/20 0.42
ALOX5 P09917 1/20 0.41
OPRM1 P35372 2/20 0.41
OPRD1 P41143 2/20 0.41
OPRK1 P41145 2/20 0.41
CHRM2 P08172 1/20 0.41
CHRM3 P20309 1/20 0.41
MEN1 O00255 3/20 0.40
KEAP1 Q14145 1/20 0.40
FKBP1A P62942 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716391 0.86 CTSD (0.43) KMT2ASIGMAR1L3MBTL1OPRK1CHRM2
SCHEMBL8715002 0.77 SIGMAR1 (0.51) SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL8713086 0.74 SLC6A4 (0.47) SIGMAR1SLC6A4
SCHEMBL8713649 0.72 OPRD1 (0.43) KMT2ASIGMAR1SLC6A4OPRM1OPRD1
SCHEMBL1838692 0.72 NPC1 (0.73) KMT2ANPC1TDP1L3MBTL1MEN1
SCHEMBL8713364 0.72 TDP1 (0.44) KMT2ASIGMAR1TDP1SLC6A4MEN1
SCHEMBL8718000 0.71 SIGMAR1 (0.46) KMT2ASIGMAR1SLC6A4OPRD1MEN1
Hydrochloric Acid SCHEMBL3086821 0.71 NPC1 (0.71) KMT2ANPC1TDP1L3MBTL1MEN1
SCHEMBL8716281 0.70 HRH4 (0.49)
SCHEMBL28208386 0.70 ALOX5 (0.57) KMT2ATDP1L3MBTL1ALOX5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0822939-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 1998-02-11 EP disclosed
WO-1996034012-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed