SCHEMBL8715002

SCHEMBL8715002

O=[C]N(C(=O)c1ccccc1)N1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.51
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
OPRD1 P41143 7/20 0.45
OPRM1 P35372 3/20 0.42
OPRK1 P41145 2/20 0.40
POLB P06746 1/20 0.40
HTR6 P50406 1/20 0.39
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
ADRB1 P08588 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713369 0.84 OPRD1 (0.49) ALDH1A1TSHROPRD1OPRM1ADRB1
SCHEMBL8713649 0.79 OPRD1 (0.43) SIGMAR1USP2ALDH1A1TSHRHSD17B10
SCHEMBL8716391 0.79 CTSD (0.43) SIGMAR1ALDH1A1TSHROPRK1HTR6
SCHEMBL8716688 0.78 HTR3E (0.50) ALDH1A1POLBHTR3EHTR3BHTR3A
SCHEMBL379431 0.77 SIGMAR1 (0.51) SIGMAR1USP2ALDH1A1TSHRHSD17B10
SCHEMBL8717153 0.77 KMT2A (0.42) SIGMAR1OPRD1OPRM1OPRK1
SCHEMBL28770204 0.76 SIGMAR1 (0.50) SIGMAR1USP2ALDH1A1TSHRHSD17B10
SCHEMBL8714113 0.75 HRH4 (0.60) ALDH1A1HSD17B10POLB
SCHEMBL16857496 0.73 CA2 (0.34)
SCHEMBL1961974 0.72 CA2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0822939-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 1998-02-11 EP disclosed
WO-1996034012-A1 CYCLIC PENTAPEPTIDE LH-RH RECEPTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed