SCHEMBL8717430

SCHEMBL8717430

Cc1ccc([C@](C)(N)CN2CC[C@H](O)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HRH1 P35367 4/20 0.36
CNR2 P34972 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
XBP1 P17861 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
OPRK1 P41145 1/20 0.34
KCNH2 Q12809 1/20 0.33
KCNA3 P22001 1/20 0.33
GRIN2B Q13224 1/20 0.33
PDCD1LG2 Q9BQ51 1/20 0.33
CD274 Q9NZQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717616 0.89 ALDH1A1 (0.37) ALDH1A1GAAKDM4EXBP1MAPK1
SCHEMBL8716993 0.89 ALDH1A1 (0.40) ALDH1A1GAAKDM4EXBP1MAPK1
SCHEMBL6425483 0.87 KCNA3 (0.44) ALDH1A1KDM4EOPRK1KCNA3
SCHEMBL8350936 0.85 ALDH1A1 (0.38) ALDH1A1GAAKDM4EHRH1CNR2
SCHEMBL8720345 0.85 OPRK1 (0.42) CNR2OPRK1
SCHEMBL8719953 0.83 ALDH1A1 (0.42) ALDH1A1HRH1SMN1; SMN2
SCHEMBL14347848 0.77 MEN1 (0.40) ALDH1A1GAAKDM4EHRH1CNR2
SCHEMBL8720326 0.77 HRH3 (0.44) ALDH1A1KDM4EHRH1SMN1; SMN2NPSR1
SCHEMBL10272308 0.72 ALDH1A1 (0.57) ALDH1A1HRH1
SCHEMBL13479261 0.72 ALDH1A1 (0.57) ALDH1A1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0569802-B1 Arylacetamides MERCK PATENT GMBH (DE) 1998-07-15 EP disclosed
EP-0569802-A1 Arylacetamides MERCK PATENT GmbH (DE) 1993-11-18 EP disclosed