SCHEMBL8717616

SCHEMBL8717616

C[C@@](N)(CN1CC[C@H](O)C1)c1ccc(N)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
XBP1 P17861 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
OPRK1 P41145 3/20 0.34
OPRM1 P35372 2/20 0.33
KCNA3 P22001 1/20 0.33
OPRD1 P41143 1/20 0.33
LTA4H P09960 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8717430 0.89 ALDH1A1 (0.37) ALDH1A1GAAKDM4EXBP1MAPK1
SCHEMBL8716993 0.89 ALDH1A1 (0.40) ALDH1A1GAAKDM4EXBP1MAPK1
SCHEMBL6425483 0.87 KCNA3 (0.44) ALDH1A1KDM4EOPRK1OPRM1KCNA3
SCHEMBL8720345 0.85 OPRK1 (0.42) OPRK1
SCHEMBL8719953 0.83 ALDH1A1 (0.42) ALDH1A1LTA4H
SCHEMBL8350936 0.74 ALDH1A1 (0.38) ALDH1A1GAAKDM4EXBP1MAPK1
SCHEMBL3935123 0.72 ALDH1A1 (0.57) ALDH1A1LTA4H
SCHEMBL3935867 0.72 ALDH1A1 (0.57) ALDH1A1LTA4H
SCHEMBL188289 0.72 ALDH1A1 (0.57) ALDH1A1LTA4H
SCHEMBL13724422 0.72 LTA4H (0.35) ALDH1A1OPRK1OPRM1KCNA3OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0569802-B1 Arylacetamides MERCK PATENT GMBH (DE) 1998-07-15 EP disclosed
EP-0569802-A1 Arylacetamides MERCK PATENT GmbH (DE) 1993-11-18 EP disclosed