SCHEMBL8720050

SCHEMBL8720050

CC(C)(C)NC(=O)OCC1CN(C(=N)N)CCO1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 12/20 0.46
NR1H4 Q96RI1 1/20 0.32
CACNA1H O95180 1/20 0.31
EPHX2 P34913 1/20 0.31
EPHA2 P29317 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24158828 0.76 PDK1 (0.63) PDK1
SCHEMBL8918034 0.76 F2 (0.38) PDK1NR1H4CACNA1HTSHR
SCHEMBL28662047 0.75 LMNA (0.42) PDK1
SCHEMBL8575864 0.73 PDK1 (0.38) PDK1
SCHEMBL17242140 0.72 ALDH1A1 (0.49) TSHR
SCHEMBL2905444 0.72 ALDH1A1 (0.49) TSHR
SCHEMBL10290412 0.72 LMNA (0.54)
SCHEMBL28091529 0.71 DRD4 (0.55)
SCHEMBL28290423 0.71 LMNA (0.49)
SCHEMBL28022537 0.70 TRPA1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763604-A ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
US-5677448-A CHEMICAL INTERMEDIATES FOR MAKING ANTAGONIST OF THROMBIN, TREATING THROMBOSIS, STROKE, INFLAMMATION, ARTERIOSCLEROSIS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1997-10-14 US disclosed