SCHEMBL8720874

SCHEMBL8720874

[N-]=[N+]=CC(=O)c1cccc(F)c1F

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.55
CES1 P23141 5/20 0.55
BCHE P06276 1/20 0.55
HPGD P15428 1/20 0.44
ALB P02768 1/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HTT P42858 1/20 0.39
HIF1A Q16665 1/20 0.39
MAOB P27338 2/20 0.38
KAT6A Q92794 1/20 0.38
ALOX15 P16050 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
ATM Q13315 1/20 0.35
GAA P10253 1/20 0.34
TDP1 Q9NUW8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9448980 0.85 CES2 (0.52) CES2CES1BCHEHPGDALDH1A1
Water SCHEMBL28342642 0.76 CES2 (0.61) CES2CES1BCHEHPGDALB
SCHEMBL3184940 0.72 CES2 (1.00) CES2CES1BCHEHPGDALB
SCHEMBL3440833 0.72 CES2 (0.74) CES2CES1BCHEHPGDALB
SCHEMBL7613879 0.72 ALDH1A1 (0.56) HPGDALDH1A1MEN1KMT2AHTT
SCHEMBL8715511 0.71 ALDH1A1 (0.42) HPGDALDH1A1MEN1KMT2AHTT
SCHEMBL9449288 0.70 CES2 (0.52) CES2CES1HPGDALDH1A1MEN1
SCHEMBL9448877 0.70 GPR52 (0.45) HPGDALDH1A1MEN1KMT2AHTT
SCHEMBL9448951 0.70 ALDH1A1 (0.46) HPGDALDH1A1MEN1KMT2AHTT
SCHEMBL31537534 0.70 CES2 (0.71) CES2CES1BCHEHPGDALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722448-A4 O-ARYL, O-ALKYL, O-ALKENYL AND O-ALKYNYL-MACROLIDES HAVING IMMUNOSUPPRESSIVE ACTIVITY MERCK & CO INC (US) 1998-04-29 EP disclosed
EP-0722448-A1 O-ARYL, O-ALKYL, O-ALKENYL AND O-ALKYNYL-MACROLIDES HAVING IMMUNOSUPPRESSIVE ACTIVITY MERCK & CO. INC. (US) 1996-07-24 EP disclosed