SCHEMBL8722135

SCHEMBL8722135

CCOC(=O)c1cnc(NC(=O)/C(=C\C=O)CN)nc1-c1ccco1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 18/20 0.48
ADORA2A P29274 18/20 0.48
ADORA1 P30542 17/20 0.48
ADORA2B P29275 9/20 0.48
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8722759 0.85 ALDH1A1 (0.55) ADORA3L3MBTL1
SCHEMBL8724476 0.83 JUN (0.44)
SCHEMBL8721300 0.82 RAB9A (0.52)
SCHEMBL8722769 0.81 JUN (0.57)
SCHEMBL8726399 0.80 RAB9A (0.42)
SCHEMBL8725171 0.80 NFKB1 (0.52)
SCHEMBL8724454 0.78 HSP90AA1 (0.55)
SCHEMBL8721318 0.77 RAB9A (0.38) ADORA3ADORA2AADORA1
SCHEMBL8721324 0.77 KDM4E (0.56) L3MBTL1
SCHEMBL8721404 0.77 NFKB1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998038171-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1998-09-03 WO disclosed
WO-1997009325-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1997-03-13 WO disclosed