SCHEMBL8722769

SCHEMBL8722769

CCOC(=O)c1cnc(NC(=O)/C(=C\C=O)CN)nc1-c1ccc(C)s1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JUN P05412 4/20 0.57
NFKB1 P19838 4/20 0.57
NFKB2 Q00653 4/20 0.57
RELA Q04206 4/20 0.57
FOS P01100 2/20 0.42
RAB9A P51151 4/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NPC1 O15118 4/20 0.39
MAPT P10636 3/20 0.39
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MPI P34949 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.35
KDM4E B2RXH2 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8724476 0.88 JUN (0.44) JUNNFKB1NFKB2RELAFOS
SCHEMBL8722759 0.85 ALDH1A1 (0.55) JUNNFKB1NFKB2RELAFOS
SCHEMBL8721300 0.84 RAB9A (0.52) JUNNFKB1NFKB2RELARAB9A
SCHEMBL8726399 0.82 RAB9A (0.42) JUNNFKB1NFKB2RELARAB9A
SCHEMBL8722135 0.81 ADORA3 (0.48)
SCHEMBL8725171 0.81 NFKB1 (0.52) JUNNFKB1NFKB2RELARAB9A
SCHEMBL8724454 0.79 HSP90AA1 (0.55) JUNNFKB1NFKB2RELARAB9A
SCHEMBL8723085 0.79 KMT2A (0.39) JUNNFKB1NFKB2RELAFOS
SCHEMBL8721318 0.79 RAB9A (0.38) JUNNFKB1NFKB2RELAFOS
SCHEMBL8721324 0.79 KDM4E (0.56) JUNNFKB1NFKB2RELAFOS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998038171-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1998-09-03 WO claimed
WO-1998038171-A1 PYRIMIDINE CARBOXYLATES AND RELATED COMPOUNDS AND METHODS FOR TREATING INFLAMMATORY CONDITIONS SIGNAL PHARMACEUTICALS, INC. (US) 1998-09-03 WO disclosed