SCHEMBL8725910

SCHEMBL8725910

O=C(O)c1cnc(CS)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALOX15 P16050 1/20 0.47
P4HA1 P13674 2/20 0.45
P4HTM Q9NXG6 2/20 0.45
HCAR2 Q8TDS4 2/20 0.44
MAPT P10636 1/20 0.44
MIF P14174 1/20 0.43
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
GABRA4 P48169 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23829753 0.77 ALDH1A1 (0.47) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL5079717 0.77 ALDH1A1 (0.47) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL186656 0.77 ALDH1A1 (0.52) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL20236440 0.77 ALDH1A1 (0.47) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL4886683 0.75 ALDH1A1 (0.58) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL27762779 0.74 ALDH1A1 (0.44) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL5660197 0.73 P4HA1 (0.56) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL10837168 0.72 HCAR3 (0.51) ALDH1A1HSD17B10KDM4EALOX15P4HA1
SCHEMBL456951 0.71 LDHA (0.46) P4HA1P4HTMMIFNAPRTHCAR3
SCHEMBL27716846 0.71 HCAR3 (0.49) ALDH1A1HSD17B10KDM4EALOX15MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873356-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-10-28 EP disclosed
WO-1996025426-A9 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS 1997-06-12 WO disclosed
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed