SCHEMBL8726250

SCHEMBL8726250

C[C@H](NC(=O)c1ccc(Oc2ccc(N(CCOS(C)(=O)=O)CCOS(C)(=O)=O)c3ccccc23)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
NPSR1 Q6W5P4 3/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA9 Q16790 2/20 0.34
MCHR1 Q99705 1/20 0.34
KEAP1 Q14145 2/20 0.33
NFE2L2 Q16236 2/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 4/20 0.33
MMP13 P45452 2/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
RECQL P46063 1/20 0.32
CACNA1H O95180 1/20 0.32
CACNA1B Q00975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726211 0.88 NPSR1 (0.37) ALDH1A1NPSR1CA12CA1CA9
SCHEMBL8726177 0.87 ALDH1A1 (0.37) ALDH1A1NPSR1POLBMAPTMEN1
SCHEMBL8726450 0.77 ALDH1A1 (0.39) ALDH1A1NPSR1POLBMAPTMEN1
SCHEMBL8722134 0.75 NPSR1 (0.44) ALDH1A1NPSR1MAPTMEN1KMT2A
SCHEMBL8724221 0.75 CA1 (0.42) ALDH1A1CA12CA1CA9MCHR1
SCHEMBL8722997 0.70 MAPT (0.37) ALDH1A1MCHR1MAPT
SCHEMBL7717390 0.70 MAPT (0.36) ALDH1A1NPSR1CA12CA1CA9
SCHEMBL8726452 0.69 MAPT (0.40) ALDH1A1NPSR1CA12CA1CA9
SCHEMBL8722158 0.68 CA2 (0.41) CA12CA1CA9KEAP1TDP1
SCHEMBL27453160 0.67 MAPT (0.54) ALDH1A1NPSR1POLBMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998035982-A1 COMPOUNDS FOR USE IN ADEPT ZENECA LIMITED (GB) 1998-08-20 WO disclosed