SCHEMBL8724221

SCHEMBL8724221

C[C@H](NC(=O)c1ccc(Oc2ccc(N(CCCl)CCCl)c3ccccc23)cc1)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
UTS2R Q9UKP6 1/20 0.40
EGFR P00533 2/20 0.38
ERBB2 P04626 2/20 0.38
BCL2L1 Q07817 1/20 0.38
MMP2 P08253 2/20 0.37
MMP9 P14780 2/20 0.37
MMP12 P39900 2/20 0.37
CA2 P00918 2/20 0.37
ESRRA P11474 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MCHR1 Q99705 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
FFAR1 O14842 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1B Q00975 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726177 0.88 ALDH1A1 (0.37) UTS2REGFRERBB2ESRRAALDH1A1
SCHEMBL8722158 0.87 CA2 (0.41) CA1CA12CA9UTS2RBCL2L1
SCHEMBL8724202 0.81 EGFR (0.43) CA1CA12CA9UTS2REGFR
SCHEMBL8722146 0.81 CA1 (0.43) CA1CA12CA9UTS2RCA2
SCHEMBL7715738 0.81 CA1 (0.44) CA1CA12CA9UTS2REGFR
SCHEMBL7715732 0.80 EGFR (0.53) CA1CA12CA9UTS2REGFR
SCHEMBL8726211 0.79 NPSR1 (0.37) CA1CA12CA9UTS2RMMP2
SCHEMBL8726250 0.75 ALDH1A1 (0.35) CA1CA12CA9ALDH1A1MCHR1
SCHEMBL8722080 0.74 MMP2 (0.55) CA1CA12CA9UTS2RMMP2
SCHEMBL8726236 0.73 TAS1R3 (0.40) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998035982-A1 COMPOUNDS FOR USE IN ADEPT ZENECA LIMITED (GB) 1998-08-20 WO disclosed