SCHEMBL8726286

SCHEMBL8726286

CCc1c(F)c(O)cc(F)c1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRB2 P07550 2/20 0.36
CYP3A4 P08684 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.35
APEX1 P27695 2/20 0.35
RECQL P46063 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
RAD52 P43351 1/20 0.35
BLM P54132 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
ESR1 P03372 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1548068 0.83 CA1 (0.33) ESR1TRPA1
SCHEMBL23492884 0.77 ESR1 (0.33) ADRB2KDM4EMAPTAPEX1RECQL
SCHEMBL12716286 0.74 RAPGEF4 (0.32)
SCHEMBL6231388 0.74 PGAM1 (0.40) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL8792389 0.73 TRPV4 (0.30)
SCHEMBL19115496 0.73 ESR1 (0.42) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL25216161 0.73 TRPA1 (0.30) TRPA1
SCHEMBL21883580 0.72 HPGD (0.41) ADRA2AADRA2CADRA1ACYP3A4HSD17B10
SCHEMBL24749310 0.71 MAPK1 (0.36) ADRA2AADRA2BADRA2CADRA1AADRB2
SCHEMBL6233326 0.71 HTT (0.50) CYP3A4KDM4EMAPTTDP1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5759956-A PYRAZINE CARBOXAMIDE DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1998-06-02 US disclosed
EP-0700391-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1996-03-13 EP disclosed
WO-1994027974-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1994-12-08 WO disclosed
EP-0038186-A2 Perfluoroamides of diaryl esters of N-phosphonomethylglycinonitrile, herbicidal compositions and herbicidal use thereof MONSANTO COMPANY (US) 1981-10-21 EP disclosed