SCHEMBL8726507

SCHEMBL8726507

C[C@H](NC(=O)c1ccc(Cc2ccc(N(CCBr)CCBr)cc2)cc1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.47
CA12 O43570 1/20 0.47
CA9 Q16790 1/20 0.47
CA2 P00918 3/20 0.45
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
LMNA P02545 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
PTGS2 P35354 1/20 0.43
PTPN1 P18031 2/20 0.42
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
CNR2 P34972 1/20 0.40
ESRRG P62508 2/20 0.39
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTT P42858 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726497 0.90 CA1 (0.49) CA1CA12CA9CA2HDAC1
SCHEMBL8726226 0.86 CA1 (0.49) CA1CA12CA9CA2LMNA
SCHEMBL8724180 0.84 CA2 (0.45) CA1CA12CA9CA2HPGD
SCHEMBL8722967 0.84 ALDH1A1 (0.41) CA1CA12CA9HDAC1HDAC6
SCHEMBL8723008 0.79 CA1 (0.42) CA1CA12CA9CA2RAB9A
SCHEMBL8721928 0.77 CA1 (0.49) CA1CA12CA9CA2HDAC1
SCHEMBL8728048 0.77 CA1 (0.40) CA1CA12CA9CA2ALDH1A1
SCHEMBL8723006 0.75 DHFR (0.33) HDAC1HDAC6LMNAALDH1A1CYP1A2
SCHEMBL8726522 0.74 CA2 (0.46) CA1CA12CA9CA2HDAC1
SCHEMBL11103451 0.74 CA2 (0.71) CA1CA12CA9CA2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998035982-A1 COMPOUNDS FOR USE IN ADEPT ZENECA LIMITED (GB) 1998-08-20 WO disclosed