SCHEMBL8728142

SCHEMBL8728142

N#Cc1cc(Cc2ccccc2)ccc1N1CCNCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.51
TAAR1 Q96RJ0 1/20 0.49
SLC6A2 P23975 2/20 0.45
SLC6A4 P31645 2/20 0.45
HTR1A P08908 2/20 0.45
SLC6A3 Q01959 1/20 0.45
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
LTA4H P09960 1/20 0.43
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
AR P10275 1/20 0.42
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
HTR2A P28223 1/20 0.41
HTR7 P34969 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL233169 0.75 ADRB1 (0.58) HTR6SLC6A2SLC6A4HTR1ASLC6A3
Hydrochloric Acid SCHEMBL20139829 0.74 ADRB1 (0.56) HTR6HTR1AALDH1A1DRD2DRD3
Hydrochloric Acid SCHEMBL29882725 0.74 ADRB1 (0.56) HTR6HTR1AALDH1A1DRD2DRD3
SCHEMBL6560078 0.74 SIGMAR1 (0.68) HTR6TAAR1SLC6A2SLC6A4HTR1A
SCHEMBL654285 0.73 ALDH1A1 (0.57) HTR6SLC6A4HTR1AALDH1A1DRD2
SCHEMBL2997329 0.73 ALDH1A1 (0.57) HTR6SLC6A2SLC6A4HTR1ASLC6A3
SCHEMBL3636287 0.73 GAA (0.56) HTR6HTR1AALDH1A1KMT2ADRD2
SCHEMBL20883839 0.73 HTR3A (0.52) HTR6TAAR1SLC6A4HTR1AALDH1A1
SCHEMBL7562266 0.73 HTR1A (0.47) SLC6A4HTR1ADRD2DRD3HTR2A
Hydrochloric Acid SCHEMBL2881381 0.72 SIGMAR1 (0.66) HTR6TAAR1SLC6A2SLC6A4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865280-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-09-23 EP disclosed
WO-1997017967-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-05-22 WO disclosed