SCHEMBL872883

SCHEMBL872883

N#CC1(C(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4)cc3)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.42
EP300 Q09472 6/20 0.41
CREBBP Q92793 6/20 0.41
PFKFB3 Q16875 12/20 0.40
PFKFB1 P16118 11/20 0.40
PFKFB2 O60825 9/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL844922 0.91 EP300 (0.48) DPP4EP300CREBBP
SCHEMBL872886 0.79 KDM4E (0.52) PFKFB3PFKFB1PFKFB2
SCHEMBL844873 0.78 NPC1 (0.63) DPP4
SCHEMBL10119687 0.78 CYP2C9 (0.44) DPP4EP300CREBBPPFKFB3PFKFB1
SCHEMBL873223 0.78 RHOC (0.43) DPP4
SCHEMBL845510 0.78 SCN3A (0.54) PFKFB3PFKFB1PFKFB2
SCHEMBL845110 0.77 ALDH1A1 (0.48) PFKFB3PFKFB1PFKFB2
SCHEMBL10119592 0.77 F2 (0.43)
SCHEMBL874324 0.77 MAPK1 (0.42) EP300CREBBP
SCHEMBL874056 0.76 TRPV1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed