SCHEMBL8733390

SCHEMBL8733390

COc1ccc(N=Nc2ccc(C(=O)Cl)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.53
CES1 P23141 2/20 0.53
CA1 P00915 5/20 0.52
CA2 P00918 5/20 0.52
HDAC1 Q13547 1/20 0.51
MAPT P10636 4/20 0.50
HPGD P15428 2/20 0.50
PTGS2 P35354 1/20 0.50
PARP1 P09874 1/20 0.50
PARP10 Q53GL7 1/20 0.50
PARP2 Q9UGN5 1/20 0.50
PARP4 Q9UKK3 1/20 0.50
ALDH1A1 P00352 2/20 0.48
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ESR1 P03372 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
TSHR P16473 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22288 0.88 CES2 (0.67) CES2CES1CA1CA2HDAC1
Hydrochloric Acid SCHEMBL27781157 0.86 CES2 (0.64) CES2CES1CA1CA2HDAC1
SCHEMBL2263327 0.84 TRPA1 (0.54) MAPTALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL2202425 0.84 TRPA1 (0.54) MAPTALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL6667738 0.82 CES2 (0.59) CES2CES1CA1CA2MAPT
SCHEMBL11511850 0.82 PARP10 (0.66) CES2CES1CA1CA2MAPT
P-Anisic Acid SCHEMBL11874860 0.81 CA1 (0.80) CES2CES1CA1CA2MAPT
SCHEMBL7722030 0.81 HPGD (0.75) CES2CES1CA1CA2MAPT
SCHEMBL11763162 0.81 ACHE (0.60) CES2CES1CA1CA2MAPT
SCHEMBL14130421 0.80 PRSS1 (0.71) CES2CES1CA1CA2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661309-B1 Use of hydroperoxide derivatives of Cyclo-olefin copolymers TICONA GMBH (DE) 1998-11-25 EP disclosed
EP-0661309-A2 Cyclo-olefin copolymers and process for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed