SCHEMBL8744690

SCHEMBL8744690

N#Cc1nc(-c2cccc(Cl)c2)c[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
CTSS P25774 1/20 0.48
CTSK P43235 1/20 0.48
ADORA2A P29274 4/20 0.48
ADORA1 P30542 4/20 0.48
ADORA2B P29275 2/20 0.48
LRRK2 Q5S007 1/20 0.46
IDO1 P14902 2/20 0.45
PDGFRB P09619 1/20 0.43
KIT P10721 1/20 0.43
KDR P35968 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
ALOX15 P16050 1/20 0.42
NUDT1 P36639 1/20 0.41
PSMB8 P28062 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
MPI P34949 1/20 0.41
GFER P55789 1/20 0.41
PLK1 P53350 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8744743 0.81 MCL1 (0.41) KDM4EADORA2AADORA1LRRK2PDGFRB
SCHEMBL7432291 0.81 ADORA2A (0.41) KDM4ECTSKADORA2AADORA1LRRK2
SCHEMBL8744764 0.81 CTSS (0.48) KDM4ECTSSCTSKADORA2AADORA1
SCHEMBL8744753 0.81 CTSS (0.49) KDM4ECTSSCTSKADORA2AADORA1
SCHEMBL8744832 0.78 MCL1 (0.42) KDM4EADORA2AADORA1ALDH1A1GAA
SCHEMBL8744699 0.77 CTSS (0.61) KDM4ECTSSCTSKIDO1ALDH1A1
SCHEMBL8744714 0.77 CTSS (0.54) CTSSCTSKLRRK2IDO1
SCHEMBL8744729 0.76 KDM4E (0.46) KDM4EPSMB8GAA
SCHEMBL8299017 0.75 PDGFRB (0.49) KDM4EIDO1PDGFRBKITKDR
SCHEMBL26112355 0.73 SCN2A (0.51) KDM4EADORA2AADORA1IDO1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed