SCHEMBL8744832

SCHEMBL8744832

N#Cc1nc(-c2ccc(-c3ccccc3)cc2)c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.42
ADORA1 P30542 3/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
ALDH1A3 P47895 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
KDM4E B2RXH2 3/20 0.40
HPGD P15428 2/20 0.40
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 3/20 0.39
ADORA2A P29274 1/20 0.39
MAPK1 P28482 1/20 0.39
MYC P01106 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CSNK1A1 P48729 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432291 0.96 ADORA2A (0.41) MCL1ADORA1CYP11B1CYP11B2KDM4E
SCHEMBL8744743 0.82 MCL1 (0.41) MCL1ADORA1KDM4EHPGDALDH1A1
SCHEMBL8744742 0.82 CYP11B1 (0.43) ADORA1CYP11B1CYP11B2KDM4EHPGD
SCHEMBL8744752 0.82 ERBB2 (0.41) ADORA1KDM4EALDH1A1ADORA2AMEN1
SCHEMBL8744693 0.80 CCNC (0.47) ADORA1ADORA2AMAPK1GSK3BRAB9A
SCHEMBL8744764 0.78 CTSS (0.48) ADORA1KDM4EHPGDALDH1A1ADORA2A
SCHEMBL8744687 0.78 KIF11 (0.47) MYC
SCHEMBL8744692 0.78 CYP2A6 (0.43) KDM4EHPGDALDH1A1MEN1KMT2A
SCHEMBL8744690 0.78 KDM4E (0.49) ADORA1KDM4EALDH1A1ADORA2AGAA
SCHEMBL8744753 0.78 CTSS (0.49) ADORA1KDM4EHPGDL3MBTL1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed