SCHEMBL8744753

SCHEMBL8744753

Cc1cccc(-c2c[nH]c(C#N)n2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.49
CTSK P43235 1/20 0.49
LRRK2 Q5S007 2/20 0.47
ADORA2A P29274 2/20 0.46
ADORA1 P30542 2/20 0.46
IDO1 P14902 1/20 0.45
METAP2 P50579 1/20 0.45
XDH P47989 1/20 0.43
ADORA2B P29275 1/20 0.40
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 2/20 0.40
AR P10275 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPK14 Q16539 1/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
KMO O15229 1/20 0.39
PIN1 Q13526 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432291 0.81 ADORA2A (0.41) CTSKLRRK2ADORA2AADORA1RAB9A
SCHEMBL8744690 0.81 KDM4E (0.49) CTSSCTSKLRRK2ADORA2AADORA1
SCHEMBL8744764 0.81 CTSS (0.48) CTSSCTSKADORA2AADORA1IDO1
SCHEMBL8744714 0.80 CTSS (0.54) CTSSCTSKLRRK2IDO1
SCHEMBL8744832 0.78 MCL1 (0.42) ADORA2AADORA1RAB9AKDM4EMAPT
SCHEMBL10604269 0.78 IDO1 (0.51) CTSSCTSKIDO1METAP2XDH
SCHEMBL8744699 0.77 CTSS (0.61) CTSSCTSKIDO1XDHKDM4E
SCHEMBL8744731 0.76 HSP90AB1 (0.45) KDM4ENPC1MAPT
SCHEMBL25357822 0.74 USP8 (0.38) LRRK2RAB9AKDM4ENPC1AR
SCHEMBL15029191 0.73 IDO1 (0.47) ADORA2AADORA1IDO1METAP2XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653421-B1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA (JP) 1997-01-15 EP disclosed
US-5552557-A Process for preparing 2-cyanoimidazole compounds by reaction of an amino ketone compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1996-09-03 US disclosed
EP-0653421-A1 Process for preparing 2-cyanoimidazole compounds ISHIHARA SANGYO KAISHA LTD. (JP) 1995-05-17 EP disclosed