SCHEMBL874617

SCHEMBL874617

O=C(Nc1ccc(-c2nc(C(F)(F)C(F)(F)F)c(C(=O)NCCN3CCCCC3)s2)cc1)c1cc2cccnc2s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
NAMPT P43490 2/20 0.43
ATR Q13535 4/20 0.39
EPHX2 P34913 3/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
KCNH2 Q12809 1/20 0.38
RAF1 P04049 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
IKBKG Q9Y6K9 1/20 0.37
JAK2 O60674 1/20 0.37
CHRNA7 P36544 3/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873629 0.84 NAMPT (0.42) DRD2DRD3NAMPTATRMKNK2
SCHEMBL874231 0.83 CHRNA7 (0.43) DRD2DRD3NAMPTCHRNA7
SCHEMBL874618 0.82 NAMPT (0.41) DRD2DRD3NAMPTCHRNA7
SCHEMBL874482 0.81 CHRM4 (0.42) DRD2DRD3NAMPTCHRNA7
SCHEMBL874535 0.81 NAMPT (0.48) DRD2DRD3NAMPTATRCYP3A4
SCHEMBL882713 0.77 CYP3A4 (0.44) DRD2DRD3NAMPTCYP3A4CYP2D6
SCHEMBL874058 0.77 NAMPT (0.42) DRD2DRD3NAMPTATRCYP3A4
SCHEMBL877180 0.76 NAMPT (0.43) DRD2DRD3NAMPTATRCYP3A4
SCHEMBL873905 0.76 DRD2 (0.48) DRD2DRD3NAMPTKCNH2CHRNA7
SCHEMBL874515 0.76 ATR (0.43) DRD2DRD3NAMPTATRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed