SCHEMBL8745797

SCHEMBL8745797

COc1ccccc1N1CCN(CCc2c(C)c3ccc(OC)c(OC)c3oc2=O)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 3/20 0.56
POLB P06746 1/20 0.56
GAA P10253 1/20 0.56
HTT P42858 1/20 0.56
ADRA1D P25100 3/20 0.51
ADRA1A P35348 3/20 0.51
ADRA1B P35368 3/20 0.51
DRD2 P14416 2/20 0.49
DRD3 P35462 2/20 0.49
HTR1A P08908 2/20 0.49
HTR2A P28223 1/20 0.49
MEN1 O00255 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
ALOX12 P18054 1/20 0.48
HTR7 P34969 1/20 0.48
KMT2A Q03164 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745810 0.90 ADRA1A (0.52) ALDH1A1KDM4EADRA1DADRA1AADRA1B
SCHEMBL8745798 0.82 BRAF (0.56) GAAADRA1DADRA1AADRA1BDRD2
SCHEMBL8745809 0.82 HTR2A (0.60) ALDH1A1KDM4EADRA1ADRD2DRD3
SCHEMBL8745769 0.79 BRAF (0.55) ALDH1A1GAAADRA1DADRA1AADRA1B
SCHEMBL6755853 0.79 KDM4E (0.62) ALDH1A1KDM4EPOLBGAAHTT
SCHEMBL8745816 0.78 ADRA1A (0.55) GAAADRA1DADRA1AADRA1BDRD2
SCHEMBL8745760 0.77 ADRA1A (0.55) GAAADRA1DADRA1AADRA1BDRD2
SCHEMBL9144743 0.77 DRD2 (0.51) ADRA1ADRD2DRD3HTR1AHTR2A
SCHEMBL8745788 0.76 ABCC1 (0.56) GAAADRA1DADRA1AADRA1BDRD2
SCHEMBL8745813 0.76 BRAF (0.49) GAAADRA1DADRA1AADRA1BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed
EP-0663911-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE. SCHWABE WILLMAR GMBH & CO (DE) 1995-07-26 EP disclosed
WO-1994008985-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1994-04-28 WO disclosed