SCHEMBL8745909

SCHEMBL8745909

Cc1ccccc1C(OC(=O)N(C)C)c1cncnc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 3/20 0.37
ITGA4 P13612 3/20 0.37
GPBAR1 Q8TDU6 3/20 0.36
ESR1 P03372 1/20 0.36
CTSA P10619 1/20 0.32
KDM4E B2RXH2 3/20 0.32
GAA P10253 2/20 0.32
CYP2D6 P10635 2/20 0.32
SLC22A2 O15244 1/20 0.32
SLC22A1 O15245 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
ADRA2A P08913 1/20 0.32
CHRM1 P11229 1/20 0.32
ADRA2B P18089 1/20 0.32
CHRM3 P20309 1/20 0.32
DRD1 P21728 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9029347 0.73 ROCK2 (0.37) GPBAR1CTSAKDM4EGAA
SCHEMBL8745964 0.69 ITGB1 (0.41) ITGB1ITGA4KDM4ECYP2D6CYP2C19
SCHEMBL8745917 0.68 HPGD (0.41) CTSAKDM4EGAACYP2C19CYP3A4
SCHEMBL9030025 0.67 GPBAR1 (0.38) GPBAR1
SCHEMBL907693 0.65 ALDH1A1 (0.39) KDM4EGAACYP2C19CYP3A4CYP2C9
SCHEMBL8828257 0.63 CASP3 (0.36) ITGB1ITGA4GPBAR1KDM4EGAA
SCHEMBL8326882 0.62 MAPT (0.40) GPBAR1GAAPOLB
SCHEMBL1838498 0.61 ESR1 (0.52) ESR1KDM4EGAACYP2D6SLC22A2
SCHEMBL8577603 0.61 GAA (0.47) ESR1GAACYP2D6CYP2C19CYP3A4
SCHEMBL11352667 0.60 RAB9A (0.41) ITGB1ITGA4GPBAR1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758323-A1 HERBICIDAL HYDROXYBENZYL-SUBSTITUTED HETEROARYL COMPOUNDS AND DERIVATIVES THEREOF ZENECA LIMITED (GB) 1997-02-19 EP disclosed