SCHEMBL8751995

SCHEMBL8751995

COc1ccnc(SCCC=C(F)F)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
MAPK1 P28482 3/20 0.35
TP53 P04637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 4/20 0.35
MAPT P10636 4/20 0.35
HSD17B10 Q99714 2/20 0.35
ADORA3 P0DMS8 2/20 0.33
ALOX15 P16050 2/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
ADORA1 P30542 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 3/20 0.32
DYRK3 O43781 1/20 0.31
DYRK1A Q13627 1/20 0.31
DYRK2 Q92630 1/20 0.31
HPGD P15428 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8752048 0.88 MAPK1 (0.32) SMN1; SMN2NPC1RAB9AMAPK1ALDH1A1
SCHEMBL8751982 0.86 NPC1 (0.31) SMN1; SMN2NPC1RAB9AMAPK1TP53
SCHEMBL8752080 0.85 ALOX15 (0.31) ALOX15KMT2A
SCHEMBL8752015 0.83 L3MBTL1 (0.33)
SCHEMBL8752040 0.83 MEN1 (0.34) MAPTKMT2AMEN1
SCHEMBL8752062 0.82 HTT (0.39) NPC1RAB9AALDH1A1MAPTKMT2A
SCHEMBL8752043 0.81 ALOX15 (0.51) SMN1; SMN2NPC1RAB9AALDH1A1MAPT
SCHEMBL8752003 0.81 ADORA3 (0.41) RAB9AMAPK1ALDH1A1HSD17B10ADORA3
SCHEMBL8752002 0.80 L3MBTL1 (0.50) SMN1; SMN2NPC1RAB9AMAPK1TP53
SCHEMBL8752023 0.80 ALDH1A1 (0.41) NPC1RAB9ANPSR1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684011-A Pyrimidine derivatives useful as nematicides ZENECA LIMITED (GB) 1997-11-04 US disclosed
EP-0660827-B1 HETEROCYCLIC COMPOUNDS WITH PARASITICAL ACTIVITY ZENECA LTD (GB) 1997-04-16 EP disclosed
EP-0660827-A1 HETEROCYCLIC COMPOUNDS WIHT PARASITICAL ACTIVITY. ZENECA LTD (GB) 1995-07-05 EP disclosed
WO-1994006777-A1 HETEROCYCLIC COMPOUNDS WIHT PARASITICAL ACTIVITY ZENECA LIMITED (GB) 1994-03-31 WO disclosed