SCHEMBL8760912

SCHEMBL8760912

CCc1c(Sc2ccccc2)n(COCC(O[SiH](C)C)C(C)(C)C)c(=O)[nH]c1=O

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8760903 0.81 ALDH1A1 (0.31) ALDH1A1TSHRMAPK1NPSR1
SCHEMBL599846 0.80 ALDH1A1 (0.41) ALDH1A1CYP2C9CYP2C19TSHRMAPK1
SCHEMBL9597854 0.78 ALDH1A1 (0.53) ALDH1A1CYP2C9CYP2C19TSHRMAPK1
SCHEMBL8760090 0.77 UPP1 (0.49) ALDH1A1CYP2C9CYP2C19TSHRMAPK1
SCHEMBL8760905 0.75 DUT (0.47) ALDH1A1CYP2C9CYP2C19TSHRMAPK1
SCHEMBL8761117 0.73 UPP1 (0.36)
SCHEMBL9353843 0.72 ALDH1A1 (0.30) ALDH1A1
SCHEMBL7259761 0.71 ALDH1A1 (0.36) ALDH1A1TSHRMAPK1NPSR1
SCHEMBL7259755 0.71 ALDH1A1 (0.34) ALDH1A1CYP2C9CYP2C19TSHRMAPK1
SCHEMBL8760122 0.71 SIRT2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449726-B1 Pyrimidine nucleoside derivative and antiviral agent containing the derivative as active ingredient MITSUBISHI CHEM CORP (JP) 1997-06-11 EP disclosed
US-5318972-A Active against retroviruses, human t-cell leukemia/lymphoma viruses MITSUBISHI KASEI CORPORATION (JP) 1994-06-07 US disclosed
EP-0449726-A1 Pyrimidine nucleoside derivative and antiviral agent containing the derivative as active ingredient Mitsubishi Chemical Corporation (JP) 1991-10-02 EP disclosed